Mahmut Gözelle
Akademisyen
- Alan
- Eczacılık Bilimi (Farmakoloji)
- Üniversite
- Gazi Üniversitesi
- Fakülte ve Bölüm
- Eczacılık Fakültesi
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Akademik Profiller
Yayınlar
- 12‐(Methyl(phenyl)amino)‐N‐(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibitionDrug Development Research2024
- 2Enzalutamide-human serum albumin interaction: Electrochemical exploration of complex formation and binding parametersMicrochemical Journal2024
- 3Linker and tail group modifications on 2-((4-isopropyl-4H-1,2,4-triazol-3-yl)thio)-N-(4-phenoxyphenyl)acetamide to improve SIRT2 inhibitory potencyFabad Journal of Pharmaceutical Sciences2024
- 4Hit evaluation results in 5-benzyl-1,3,4-thiadiazole-2-carboxamide based SIRT2-selective inhibitor with improved affinity and selectivityBioorganic Chemistry2022
- 5The potential of 4-aryl-6-morpholino-3(2H)-pyridazinone-2-arylpiperazinylacetamide as a new scaffold for SIRT2 inhibition: in silico approach guided by pharmacophore mapping and molecular dockingMedicinal Chemistry Research2021
- 6Hit-to-lead optimization on aryloxybenzamide derivative virtual screening hit against SIRTBioorganic & Medicinal Chemistry2021
- 7Pharmacophore modeling and virtual screening studies to identify novel selective SIRT2 inhibitorsJournal of Molecular Graphics and Modelling2019
- 82019
- 9Structure-based exploration and pharmacological evaluation of N-substituted piperidin-4-yl-methanamine CXCR4 chemokine receptor antagonistsEuropean Journal of Medicinal Chemistry2019
- 10Synthesis, crystal structure, spectroscopic and density functional modelling studies of the 2-isopropylbenzimidazolium tetrachloroplatinate(II) monohydrateGazi University Journal of Science2017
Yayın listesi ORCID kaydından alındı.